Polycyclic Sulfoximines as New Scaffolds for Drug Discovery


[1]

0 0
  • M.L.G. Borst, C.M.J. Ouairy, S.C. Fokkema, A. Cecchi, J.M.C.A. Kerckhoffs, V.L. de Boer, P.J. van den Boogaard, R.F. Bus, R. Ebens, R. van der Hulst, J. Knol, R. Libbers, Z.M. Lion, B.W. Settels, E. de Wever, K.A. Attia, P. Sinnema, J.M. de Gooijer, K. Harkema, M. Hazewinkel, S. Snijder, and K. Pouwer, "Polycyclic Sulfoximines as New Scaffolds for Drug Discovery", ACS Combinatorial Science, vol. 20, pp. 335-343, 2018. http://dx.doi.org/10.1021/acscombsci.7b00150
  • Elucidating the Role of the Boronic Esters in the Suzuki–Miyaura Reaction: Structural, Kinetic, and Computational Investigations

    from the Scott E. Denmark group

    [1]

    0 0
  • A.A. Thomas, A.F. Zahrt, C.P. Delaney, and S.E. Denmark, "Elucidating the Role of the Boronic Esters in the Suzuki–Miyaura Reaction: Structural, Kinetic, and Computational Investigations", Journal of the American Chemical Society, vol. 140, pp. 4401-4416, 2018. http://dx.doi.org/10.1021/jacs.8b00400
  • A platform for automated nanomole-scale reaction screening and micromole-scale synthesis in flow

    [Pfizer]

    [1]

    0 0
  • D. Perera, J.W. Tucker, S. Brahmbhatt, C.J. Helal, A. Chong, W. Farrell, P. Richardson, and N.W. Sach, "A platform for automated nanomole-scale reaction screening and micromole-scale synthesis in flow", Science, vol. 359, pp. 429-434, 2018. http://dx.doi.org/10.1126/science.aap9112
  • Esterification of Carboxylic Acids with Difluoromethyl Diazomethane and Interrupted Esterification with Trifluoromethyl Diazomethane: A Fluorine Effect


    [1]

    0 0
  • S. Peng, X. Zhang, L. Zhang, and X. Hu, "Esterification of Carboxylic Acids with Difluoromethyl Diazomethane and Interrupted Esterification with Trifluoromethyl Diazomethane: A Fluorine Effect", Organic Letters, vol. 19, pp. 5689-5692, 2017. http://dx.doi.org/10.1021/acs.orglett.7b02866
  • Exploiting a “Beast” in Carbenoid Chemistry: Development of a Straightforward Direct Nucleophilic Fluoromethylation Strategy


    [1]

    0 0
  • G. Parisi, M. Colella, S. Monticelli, G. Romanazzi, W. Holzer, T. Langer, L. Degennaro, V. Pace, and R. Luisi, "Exploiting a “Beast” in Carbenoid Chemistry: Development of a Straightforward Direct Nucleophilic Fluoromethylation Strategy", Journal of the American Chemical Society, vol. 139, pp. 13648-13651, 2017. http://dx.doi.org/10.1021/jacs.7b07891