Mois : novembre 2019

Electrophotocatalytic SNAr Reactions of Unactivated Aryl Fluorides at Ambient Temperature and Without BaseElectrophotocatalytic SNAr Reactions of Unactivated Aryl Fluorides at Ambient Temperature and Without Base

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  • H. Huang, and T.H. Lambert, "Electrophotocatalytic S N Ar Reactions of Unactivated Aryl Fluorides at Ambient Temperature and Without Base", Angewandte Chemie International Edition, vol. 59, pp. 658-662, 2020. http://dx.doi.org/10.1002/anie.201909983
  • Direct Use of Carboxylic Acids in the Photocatalytic Hydroacylation of Styrenes To Generate Dialkyl Ketones

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  • J.I. Martinez Alvarado, A.B. Ertel, A. Stegner, E.E. Stache, and A.G. Doyle, "Direct Use of Carboxylic Acids in the Photocatalytic Hydroacylation of Styrenes To Generate Dialkyl Ketones", Organic Letters, vol. 21, pp. 9940-9944, 2019. http://dx.doi.org/10.1021/acs.orglett.9b03871
  • Nitroacetic Esters in the Regioselective Synthesis of Isoxazole-3,5-dicarboxylic Acid Derivatives

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  • A.Y. Smirnov, E.R. Zaitseva, O.A. Belozerova, R.S. Alekseyev, N.S. Baleeva, M.B. Zagudaylova, A.A. Mikhaylov, and M.S. Baranov, "Nitroacetic Esters in the Regioselective Synthesis of Isoxazole-3,5-dicarboxylic Acid Derivatives", The Journal of Organic Chemistry, vol. 84, pp. 15417-15428, 2019. http://dx.doi.org/10.1021/acs.joc.9b02427
  • Site‐Selective, Modular Diversification of Polyhalogenated Aryl Fluorosulfates (ArOSO2F) Enabled by an Air‐Stable Pd(I) Dimer

    Very interesting solvent effect described by Schoenebeck, making it possible to selectively couple @ C-Br, then @ C-OSO2F, and finally @ C-Cl bonds on a range of substrates.
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  • M. Mendel, I. Kalvet, D. Hupperich, G. Magnin, and F. Schoenebeck, "Site‐Selective, Modular Diversification of Polyhalogenated Aryl Fluorosulfates (ArOSO 2 F) Enabled by an Air‐Stable Pd I Dimer", Angewandte Chemie International Edition, vol. 59, pp. 2115-2119, 2020. http://dx.doi.org/10.1002/anie.201911465
  • Immunity-Guided Identification of Threonyl-tRNA Synthetase as the Molecular Target of Obafluorin, a ß-Lactone Antibiotic

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  • T.A. Scott, S.F.D. Batey, P. Wiencek, G. Chandra, S. Alt, C.S. Francklyn, and B. Wilkinson, "Immunity-Guided Identification of Threonyl-tRNA Synthetase as the Molecular Target of Obafluorin, a β-Lactone Antibiotic", ACS Chemical Biology, vol. 14, pp. 2663-2671, 2019. http://dx.doi.org/10.1021/acschembio.9b00590
  • Discovery of BAY-298 and BAY-899: Tetrahydro-1,6-naphthyridine-Based, Potent, and Selective Antagonists of the Luteinizing Hormone Receptor Which Reduce Sex Hormone Levels in Vivo

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  • L. Wortmann, B. Lindenthal, P. Muhn, A. Walter, R. Nubbemeyer, D. Heldmann, L. Sobek, F. Morandi, A.K. Schrey, D. Moosmayer, J. Günther, J. Kuhnke, M. Koppitz, U. Lücking, U. Röhn, M. Schäfer, K. Nowak-Reppel, R. Kühne, H. Weinmann, and G. Langer, "Discovery of BAY-298 and BAY-899: Tetrahydro-1,6-naphthyridine-Based, Potent, and Selective Antagonists of the Luteinizing Hormone Receptor Which Reduce Sex Hormone Levels in Vivo", Journal of Medicinal Chemistry, vol. 62, pp. 10321-10341, 2019. http://dx.doi.org/10.1021/acs.jmedchem.9b01382