An unusual bioisostere phenyl


  • Y. Wang, H. Zhao, J.T. Brewer, H. Li, Y. Lao, W. Amberg, B. Behl, I. Akritopoulou-Zanze, J. Dietrich, U.E.W. Lange, F. Pohlki, C. Hoft, W. Hornberger, S.W. Djuric, J. Sydor, M. Mezler, A.L. Relo, and A. Vasudevan, "De Novo Design, Synthesis, and Biological Evaluation of 3,4-Disubstituted Pyrrolidine Sulfonamides as Potent and Selective Glycine Transporter 1 Competitive Inhibitors", Journal of Medicinal Chemistry, vol. 61, pp. 7486-7502, 2018.

  • [1]

  • M.L.G. Borst, C.M.J. Ouairy, S.C. Fokkema, A. Cecchi, J.M.C.A. Kerckhoffs, V.L. de Boer, P.J. van den Boogaard, R.F. Bus, R. Ebens, R. van der Hulst, J. Knol, R. Libbers, Z.M. Lion, B.W. Settels, E. de Wever, K.A. Attia, P. Sinnema, J.M. de Gooijer, K. Harkema, M. Hazewinkel, S. Snijder, and K. Pouwer, "Polycyclic Sulfoximines as New Scaffolds for Drug Discovery", ACS Combinatorial Science, vol. 20, pp. 335-343, 2018.
  • from the Scott E. Denmark group


  • A.A. Thomas, A.F. Zahrt, C.P. Delaney, and S.E. Denmark, "Elucidating the Role of the Boronic Esters in the Suzuki–Miyaura Reaction: Structural, Kinetic, and Computational Investigations", Journal of the American Chemical Society, vol. 140, pp. 4401-4416, 2018.