[1]

  • A. Ochen, R. Whitten, H.E. Aylott, K. Ruffell, G.D. Williams, F. Slater, A. Roberts, P. Evans, J.E. Steves, and M.J. Sanganee, "Development of a Large-Scale Copper(I)/TEMPO-Catalyzed Aerobic Alcohol Oxidation for the Synthesis of LSD1 Inhibitor GSK2879552", Organometallics, vol. 38, pp. 176-184, 2018. http://dx.doi.org/10.1021/acs.organomet.8b00546
  • An unusual bioisostere phenyl

    [1]

  • Y. Wang, H. Zhao, J.T. Brewer, H. Li, Y. Lao, W. Amberg, B. Behl, I. Akritopoulou-Zanze, J. Dietrich, U.E.W. Lange, F. Pohlki, C. Hoft, W. Hornberger, S.W. Djuric, J. Sydor, M. Mezler, A.L. Relo, and A. Vasudevan, "De Novo Design, Synthesis, and Biological Evaluation of 3,4-Disubstituted Pyrrolidine Sulfonamides as Potent and Selective Glycine Transporter 1 Competitive Inhibitors", Journal of Medicinal Chemistry, vol. 61, pp. 7486-7502, 2018. http://dx.doi.org/10.1021/acs.jmedchem.8b00295

  • [1]

  • M.L.G. Borst, C.M.J. Ouairy, S.C. Fokkema, A. Cecchi, J.M.C.A. Kerckhoffs, V.L. de Boer, P.J. van den Boogaard, R.F. Bus, R. Ebens, R. van der Hulst, J. Knol, R. Libbers, Z.M. Lion, B.W. Settels, E. de Wever, K.A. Attia, P. Sinnema, J.M. de Gooijer, K. Harkema, M. Hazewinkel, S. Snijder, and K. Pouwer, "Polycyclic Sulfoximines as New Scaffolds for Drug Discovery", ACS Combinatorial Science, vol. 20, pp. 335-343, 2018. http://dx.doi.org/10.1021/acscombsci.7b00150